BDBM381326 4-Chloro-1-(4-methoxy-butyl)-3- methyl-1H-pyrazolo[3,4- b]pyridine-5-carboxylic acid (4- trifluoromethyl-phenyl)-amide::US10272074, Example 159
SMILES COCCCCn1nc(C)c2c(Cl)c(cnc12)C(=O)Nc1ccc(cc1)C(F)(F)F
InChI Key InChIKey=RLUJEOIHFXXLKQ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 381326
TargetGlucocorticoid receptor(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute
US Patent
Sanford Burnham Prebys Medical Discovery Institute
US Patent
Affinity DataIC50: <50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair