BDBM383504 US10280149, Example 9::[(3R)-1-cyclopentyl-3-piperidyl]-(6-methoxy-2-naphthyl)methanone

SMILES COc1ccc2cc(ccc2c1)C(=O)[C@@H]3CCCN(C3)C4CCCC4

InChI Key InChIKey=JNSVKSRNLAOUJI-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 383504   

TargetLysine-specific demethylase 2B(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 383504BDBM383504([(3R)-1-cyclopentyl-3-piperidyl]-(6-methoxy-2-naph...)
Affinity DataIC50: 3.00E+3nMAssay Description:Full length KDM2B was cloned, expressed, and purified to homogeneity. Compound inhibition of KDM2B demethylase activity was assessed by monitoring th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2020
Entry Details
US Patent