BDBM4201 2-(2,6-dioxopiperidin-3-yl)-4-((5-(3-fluoro- 4-methoxyphenyl)-1-methyl-1H- benzo[d]imidazol-6-yl)amino)isoindoline- 1,3-dione::US20240208937, Compound 5

SMILES COc1ccc(-c2cc3ncn(C)c3cc2Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1F

InChI Key InChIKey=KVWCBPNVVCHGEW-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 4201   

TargetProtein Wiz(Homo sapiens)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 4201BDBM4201(2-(2,6-dioxopiperidin-3-yl)-4-((5-(3-fluoro- 4-met...)
Affinity DataEC50:  55nMAssay Description:The kinase activity was determined by quantitation of the amount of radioactive phosphate transferred to myelin basic protein (MBP) with or without i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent

TargetZinc finger and BTB domain-containing protein 7A(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 4201BDBM4201(2-(2,6-dioxopiperidin-3-yl)-4-((5-(3-fluoro- 4-met...)
Affinity DataEC50:  55nMAssay Description:The kinase activity was determined by quantitation of the amount of radioactive phosphate transferred to myelin basic protein (MBP) with or without i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent