BDBM456055 US10723709, Example 5
SMILES CN1CCN(CC1)c1nc(c(F)s1)-c1ccc(cc1)C(=O)NC(C=O)(C1CCCC1)N1CC(C#C)C2OCC(=O)C12
InChI Key InChIKey=CSNLQUVWWAGDSS-UHFFFAOYSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 456055
Affinity DataKi: 0.600nMAssay Description:The recombinant cathepsin K can be expressed in a variety of commercially available expression systems including E coli, Pichia and Baculovirus syste...More data for this Ligand-Target Pair
Affinity DataKi: 1.17E+3nMAssay Description:The enzyme is commercially available human cathepsin L. The substrate is H-D-Val-Leu-Lys-AMC available from Bahcem. The assay buffer is 100 mM sodium...More data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:The assay uses baculovirus-expressed human cathepsin S and the boc-Val-Leu-Lys-AMC fluorescent substrate available from Bachem in a 384 well plate fo...More data for this Ligand-Target Pair