BDBM458124 US10752616, Code No. BHBA-003

SMILES Cc1ccc(C)c2oc(cc12)-c1nc(no1)-c1ccc(cc1Br)C(O)=O

InChI Key InChIKey=WHLJYGPLQBZWJL-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 458124   

TargetRetinoic acid receptor beta(Human)
King''S College London

US Patent
LigandPNGBDBM458124(US10752616, Code No. BHBA-003)
Affinity DataEC50:  16nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2021
Entry Details
US Patent

TargetRetinoic acid receptor gamma(Human)
King''S College London

US Patent
LigandPNGBDBM458124(US10752616, Code No. BHBA-003)
Affinity DataEC50:  36nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2021
Entry Details
US Patent

TargetRetinoic acid receptor alpha(Human)
King''S College London

US Patent
LigandPNGBDBM458124(US10752616, Code No. BHBA-003)
Affinity DataEC50:  160nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2021
Entry Details
US Patent