BDBM47276 US9018217, 1-Methyl-3-(2-[2-[2-(5-methyl-[1,2,4]triazolo[1,5-a]pyridin-2-yl)-ethyl]-4-phenyl-imidazol-1-yl)-ethyl)-imidazolidin-2-one::US9592230, 8-Methyl-2-{2-[1-(2-morpholin-4-yl-ethyl)-4-phenyl-1H-imidazol-2-yl]-ethyl}-[1,2,4]triazolo[1,5-a]pyridine

SMILES Cc1cccn2nc(CCc3nc(cn3CCN3CCOCC3)-c3ccccc3)nc12

InChI Key InChIKey=GYQBWMQAVCGPTB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 47276   

LigandPNGBDBM47276(US9018217, 1-Methyl-3-(2-[2-[2-(5-methyl-[1,2,4]tr...)
Affinity DataIC50: 8.10nMAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2019
Entry Details
US Patent

LigandPNGBDBM47276(US9018217, 1-Methyl-3-(2-[2-[2-(5-methyl-[1,2,4]tr...)
Affinity DataIC50: 8.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
US Patent