BDBM47285 US9018217, 1-(2-[2-[2-(5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-ethyl]-4-phenyl-imidazol-1-yl}-ethyl)-3-methyl-imidazolidin-2-one::US9592230, 1-(2-[2-[2-(5,7-Dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)-ethyl]-4-phenyl-imidazol-1-yl}-ethyl)-3-methyl-imidazolidin-2-one

SMILES CN1CCN(CCn2cc(nc2CCc2nc3nc(C)cc(C)n3n2)-c2ccccc2)C1=O

InChI Key InChIKey=BOVVUYOCMYGSHB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 47285   

LigandPNGBDBM47285(US9018217, 1-(2-[2-[2-(5,7-Dimethyl-[1,2,4]triazol...)
Affinity DataIC50: 4.40nMAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2019
Entry Details
US Patent

LigandPNGBDBM47285(US9018217, 1-(2-[2-[2-(5,7-Dimethyl-[1,2,4]triazol...)
Affinity DataIC50: 4.40nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2015
Entry Details
US Patent