BDBM4847 2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-6- (tetrahydro-2H-pyran-4-yl)-1H-indazol-5- yl)amino)isoindoline-1,3-dione::US20240208937, Compound 22

SMILES Cn1ncc2cc(Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)c(C3CCOCC3)cc21

InChI Key InChIKey=GCAPJPHGEKRMHF-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 4847   

TargetProtein Wiz(Homo sapiens)
Bristol Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 4847BDBM4847(2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-6- (tetra...)
Affinity DataEC50:  55nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent

TargetZinc finger and BTB domain-containing protein 7A(Human)
Bristol Myers Squibb

US Patent
LigandChemical structure of BindingDB Monomer ID 4847BDBM4847(2-(2,6-dioxopiperidin-3-yl)-4-((1-methyl-6- (tetra...)
Affinity DataEC50: >100nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent