BDBM495036 US10995084, Ex. No. 1A-2
SMILES Cc1cc(Cc2ccc(cc2C)C(=O)NCC(=O)N2[C@@H](CC[C@@H]2C(C)(C)C#N)c2cccc(F)c2)c(=O)[nH]n1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 495036
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Kissei Pharmaceutical
US Patent
Kissei Pharmaceutical
US Patent
Affinity DataKi: 0.0600nMAssay Description:The binding affinity assay of compounds for human CGRP receptor was carried out by inhibition of radiolabeled ligand [125I]-CGRP binding in human neu...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Kissei Pharmaceutical
US Patent
Kissei Pharmaceutical
US Patent
Affinity DataIC50: 0.120nMAssay Description:The binding affinity assay of compounds for human CGRP receptor was carried out by inhibition of radiolabeled ligand [125I]-CGRP binding in human neu...More data for this Ligand-Target Pair