BDBM495145 US10995084, Ex. No. 5A-7
SMILES CCC(C)(C)[C@H]1CC[C@H](N1C(=O)CNC(=O)c1ccc(Cc2cc(C)n[nH]c2=O)c(C)c1)c1cccc(F)c1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 495145
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Kissei Pharmaceutical
US Patent
Kissei Pharmaceutical
US Patent
Affinity DataKi: 0.0500nMAssay Description:The binding affinity assay of compounds for human CGRP receptor was carried out by inhibition of radiolabeled ligand [125I]-CGRP binding in human neu...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Kissei Pharmaceutical
US Patent
Kissei Pharmaceutical
US Patent
Affinity DataIC50: 1.10nMAssay Description:The binding affinity assay of compounds for human CGRP receptor was carried out by inhibition of radiolabeled ligand [125I]-CGRP binding in human neu...More data for this Ligand-Target Pair