BDBM4975 cid_6035592

SMILES Cc1cc(-c2cc3c(cc2Nc2cccc4c2C(=O)N(C2CCC(=O)NC2=O)C4=O)nc(C)n3C)ccn1

InChI Key InChIKey=GMKABSSSWHQPRP-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 4975   

TargetProtein Wiz(Homo sapiens)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 4975BDBM4975(4-((1,2-dimethyl-6-(2-methylpyridin-4-yl)- 1H-benz...)
Affinity DataEC50: <10nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent

TargetZinc finger and BTB domain-containing protein 7A(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 4975BDBM4975(4-((1,2-dimethyl-6-(2-methylpyridin-4-yl)- 1H-benz...)
Affinity DataEC50: >100nMAssay Description:The HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase acti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2026
Entry Details
US Patent