BDBM50004336 CHEMBL3237853
SMILES Cc1nn(C)c2nnc(Nc3ccc(cc3)S(=O)(=O)N3CCCCC3)nc12
InChI Key InChIKey=LIVSCLDRZBLHMQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50004336
TargetCarbonic anhydrase 12(Human)
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Inhibition of human carbonic anhydrase 12-mediated CO2 hydration preincubated for 15 mins by stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 2(Human)
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Affinity DataKi: 492nMAssay Description:Inhibition of human carbonic anhydrase 2-mediated CO2 hydration preincubated for 15 mins by stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Human)
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human carbonic anhydrase 1-mediated CO2 hydration preincubated for 15 mins by stopped-flow assayMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 9(Human)
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of human carbonic anhydrase 9-mediated CO2 hydration preincubated for 15 mins by stopped-flow assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Human)
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of recombinant Abl kinase (unknown origin) expressed in Sf9 cells using GGEAIYAAPFKK as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in Sf9 cells using histone H1 as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Human)
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Siedlce University of Natural Sciences and Humanities
Curated by ChEMBL
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CK2alpha1 (unknown origin) using casein as substrate in presence of [gamma33P]ATPMore data for this Ligand-Target Pair