BDBM50007562 4-{4-[2-(4-Naphthalen-1-yl-piperazin-1-yl)-ethyl]-phenyl}-thiazol-2-ylamine::CHEMBL300849

SMILES Nc1nc(cs1)-c1ccc(CCN2CCN(CC2)c2cccc3ccccc23)cc1

InChI Key InChIKey=IHLXCIWXJLTTDK-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50007562   

Target5-hydroxytryptamine receptor 1A(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50007562(CHEMBL300849 | 4-{4-[2-(4-Naphthalen-1-yl-piperazi...)
Affinity DataIC50: 11nMAssay Description:Binding affinity to 5-hydroxytryptamine 1A receptor in the rat brain using [3H]8-hydroxy-2-(di-n-propylamine)tetralin as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50007562(CHEMBL300849 | 4-{4-[2-(4-Naphthalen-1-yl-piperazi...)
Affinity DataIC50: 72nMAssay Description:Binding affinity to dopamine receptor D2 in the rat brain using [3H]NPA as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed