BDBM50011631 2-{3-[6-(2-Fluoro-phenyl)-1-trifluoromethyl-4H-2,3,5,10b-tetraaza-benzo[e]azulen-8-yl]-prop-2-ynyl}-isoindole-1,3-dione::CHEMBL20194

SMILES Fc1ccccc1C1=NCc2nnc(n2-c2ccc(cc12)C#CCN1C(=O)c2ccccc2C1=O)C(F)(F)F

InChI Key InChIKey=BEZCSEHUPFTOSA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50011631   

TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011631(CHEMBL20194 | 2-{3-[6-(2-Fluoro-phenyl)-1-trifluor...)
Affinity DataIC50: 5nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed