BDBM50018287 (R)-{3-[(Naphthalene-2-carbonyl)-amino]-2-oxo-2,3,4,5-tetrahydro-benzo[b]azepin-1-yl}-acetic acid tert-butyl ester::CHEMBL297534::{3-[(Naphthalene-2-carbonyl)-amino]-2-oxo-2,3,4,5-tetrahydro-benzo[b]azepin-1-yl}-acetic acid tert-butyl ester

SMILES CC(C)(C)OC(=O)CN1c2ccccc2CCC(NC(=O)c2ccc3ccccc3c2)C1=O

InChI Key InChIKey=QYPQPHZJHKGOLX-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50018287   

TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50018287(CHEMBL297534 | {3-[(Naphthalene-2-carbonyl)-amino]...)
Affinity DataIC50: 7.5nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50018287(CHEMBL297534 | {3-[(Naphthalene-2-carbonyl)-amino]...)
Affinity DataIC50: 7.5nMAssay Description:Ability to inhibit the binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50018287(CHEMBL297534 | {3-[(Naphthalene-2-carbonyl)-amino]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to inhibit the binding of [125I]CCK-8 to Cholecystokinin type B receptor in guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article