BDBM50019522 CHEMBL3291077

SMILES COc1cc2C(=O)N(CCCN3CCCCC3)Cc3cccc(n1)c23

InChI Key InChIKey=LVUVZVOZLPYXEO-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50019522   

Target5-hydroxytryptamine receptor 4(Guinea pig)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50019522(CHEMBL3291077)
Affinity DataKi:  283nMAssay Description:Displacement of [3H]GR113808 from Dunkin-Hartley guinea pig brain striatum 5HT4R after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50019522(CHEMBL3291077)
Affinity DataIC50: 916nMAssay Description:Antagonist activity at Rluc-tagged human 5HT4R expressed in human SH-SY5Y cells assessed as inhibition of serotonin-induced receptor/Gbeta1 coupling ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed