BDBM50025024 CHEMBL3337850
SMILES CN(C)c1cc(ccn1)C(=O)Nc1nc2cc3OC(F)(F)Oc3cc2[nH]1
InChI Key InChIKey=VCOIFZFTTRCGTJ-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50025024
Affinity DataIC50: 420nMAssay Description:Inhibition of human recombinant CK1epsilon expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital
Curated by ChEMBL
Ulm University Hospital
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of rat CK1delta kinetic domain expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital
Curated by ChEMBL
Ulm University Hospital
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of GST-tagged rat CK1delta expressed in Escherichia coli using GST-p53 (1 to 64 residues) by SDS-PAGE based autoradiographyMore data for this Ligand-Target Pair