BDBM50034467 2-Amino-N-[4-(3,4-dimethyl-isoxazol-5-ylsulfamoyl)-phenyl]-acetamide::CHEMBL26470

SMILES Cc1noc(NS(=O)(=O)c2ccc(NC(=O)CN)cc2)c1C

InChI Key InChIKey=KYXIMAVSGGCUAG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50034467   

TargetEndothelin-1 receptor(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50034467(2-Amino-N-[4-(3,4-dimethyl-isoxazol-5-ylsulfamoyl)...)
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonism of [125 I]ET-1 binding to the rat endothelin receptor in vascular smooth muscle VSM-A10 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed