BDBM50036525 CHEMBL3353569

SMILES FC(F)(F)c1cnc(N(Cc2ccccc2)S(=O)(=O)c2ccccc2)c(Cl)c1

InChI Key InChIKey=YIXMUAOMXLAEIN-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50036525   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Raqualia Pharma

Curated by ChEMBL

LigandBDBM50036525(CHEMBL3353569)Copy SMILESCopy InChI

Affinity DataIC50: 183nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as inhibition of menthol induced Ca2+ influxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
3/15/2016
Entry Details Article
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