BDBM50046399 CHEMBL3314413

SMILES CSC(=O)NCCc1c[nH]c2ccccc12

InChI Key InChIKey=UFBJIWZJGBIRMB-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50046399   

TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rat)
Vietnam Academy of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50046399(CHEMBL3314413)
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rat)
Vietnam Academy of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50046399(CHEMBL3314413)
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-intact Wistar rat aorta rings assessed as relaxation of 30 mM K+-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rat)
Vietnam Academy of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50046399(CHEMBL3314413)
Affinity DataIC50: 7.94E+4nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of 60 mM K+-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C/alpha-1D/alpha-1S(Rat)
Vietnam Academy of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50046399(CHEMBL3314413)
Affinity DataIC50: 1.26E+5nMAssay Description:Inhibition of L-type calcium channel in endothelium-denuded Wistar rat aorta rings assessed as relaxation of 30 mM K+-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2016
Entry Details Article
PubMed