BDBM50063315 CHEMBL3398446
SMILES Cc1oc(nc1CCOc1cccc(C[C@@H]2CN(C[C@@H]2C(O)=O)c2nccc(n2)C(F)(F)F)c1)-c1ccccc1
InChI Key InChIKey=CIUUZBXRQNCUIL-GGAORHGYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50063315
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Binding affinity to PPARgamma (unknown origin) using fluorescein-tagged dual PPARalpha/gamma activator by homogeneous fluorescence polarization bindi...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at GAL4 tagged human PPARalpha ligand binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Binding affinity to PPARalpha (unknown origin) using fluorescein-tagged dual PPARalpha/gamma activator by homogeneous fluorescence polarization bindi...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Bristol-Myers Squibb Research And Development (R & D)
Curated by ChEMBL
Affinity DataEC50: 2.50E+3nMAssay Description:Agonist activity at GAL4 tagged human PPARgamma ligand binding domain expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair