BDBM50086720 CHEMBL3426358

SMILES CN(C)c1ccc(\C=C\c2nc3cc(ccc3[nH]2)-c2ccccc2NS(C)(=O)=O)cc1

InChI Key InChIKey=GRUYEJOLVKNPLX-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50086720   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
TBA

Curated by ChEMBL

LigandBDBM50086720(CHEMBL3426358)Copy SMILESCopy InChI

Affinity DataIC50: 240nMAssay Description:Antagonist activity at recombinant human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced Ca2+ influx preincubated for 5 m...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/6/2016
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL