BDBM50086731 CHEMBL3426343

SMILES CC(C)(C)OC(=O)Nc1ccccc1-c1ccc2[nH]c(\C=C\c3ccc(cc3)C(C)(C)C)nc2c1

InChI Key InChIKey=NWCRPUDZGTWWAP-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50086731   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
TBA

Curated by ChEMBL

LigandBDBM50086731(CHEMBL3426343)Copy SMILESCopy InChI

Affinity DataIC50: 280nMAssay Description:Antagonist activity at recombinant human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced Ca2+ influx preincubated for 5 m...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/6/2016
Entry Details Article
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