BDBM50086735 CHEMBL3426337

SMILES CC(C)(C)c1ccc(\C=C\c2nc3cc(ccc3[nH]2)-c2ccccc2C(N)=O)cc1

InChI Key InChIKey=JAWYCUCOUVBJQW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50086735   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
TBA

Curated by ChEMBL

LigandBDBM50086735(CHEMBL3426337)Copy SMILESCopy InChI

Affinity DataIC50: 40nMAssay Description:Antagonist activity at recombinant human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced Ca2+ influx preincubated for 5 m...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/6/2016
Entry Details Article
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