BDBM50086866 CHEMBL3426365

SMILES CC(C)(O)c1ccccc1-c1ccc2[nH]c(\C=C\c3ccc(cc3)S(=O)(=O)C(F)(F)F)nc2c1

InChI Key InChIKey=ZJMZJFZVCIVNBL-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50086866   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
TBA

Curated by ChEMBL

LigandBDBM50086866(CHEMBL3426365)Copy SMILESCopy InChI

Affinity DataIC50: 19nMAssay Description:Antagonist activity at recombinant human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced Ca2+ influx preincubated for 5 m...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
5/6/2016
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL