BDBM50088023 CHEMBL3427118

SMILES CC1CCN(CC1)c1nc(ccc1CNC(=O)C(C)(C)c1ccc(NS(C)(=O)=O)c(F)c1)C(F)(F)F

InChI Key InChIKey=XCUBPGSXTUDSLA-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50088023   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50088023(CHEMBL3427118)
Affinity DataKi:  49nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced activation by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2016
Entry Details Article
PubMed