BDBM50088140 CHEMBL3427231::US9365511, 8

SMILES C[C@@H]1CCCN1CCc1ccc(cc1)-c1ccc(CCn2ncnn2)cc1

InChI Key InChIKey=XKUCBPWVGMSFND-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50088140   

TargetHistamine H3 receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088140(CHEMBL3427231 | US9365511, 8)
Affinity DataIC50: 1.20nMAssay Description:Compounds of the present invention were evaluated using the human H3 receptor (H3R) HTRF cAMP assay. In this assay, HEK293 cells expressing the human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetHistamine H3 receptor(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM50088140(CHEMBL3427231 | US9365511, 8)
Affinity DataIC50: 1.20nMAssay Description:Modulation of human histamine H3 receptor expressed in HEK293 cells assessed as change in forskolin-stimulated cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2016
Entry Details Article
PubMed