BDBM50092625 3-[3-Iodo-5-(3-trifluoromethyl-3H-diazirin-3-yl)-benzyl]-5-phenyl-3,5-dihydro-1,3,5,6-tetraaza-cyclopenta[a]naphthalen-4-one::CHEMBL340379

SMILES FC(F)(F)C1(N=N1)c1cc(I)cc(Cn2cnc3c2c(=O)n(-c2ccccc2)c2ncccc32)c1

InChI Key InChIKey=RNMWWEZUYMOMIS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50092625   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50092625(3-[3-Iodo-5-(3-trifluoromethyl-3H-diazirin-3-yl)-b...)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human PDE4A expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed