BDBM50092683 CHEMBL126366::N,N-Diethyl-4-(isoquinolin-5-yl-piperazin-1-yl-methyl)-benzamide
SMILES CCN(CC)C(=O)c1ccc(cc1)C(N1CCNCC1)c1cccc2cnccc12
InChI Key InChIKey=WAXHVFCFNPHKLK-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50092683
Affinity DataEC50: 55nMAssay Description:Agonist potency was measured using GTP gamma-[35S] binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against cloned human Opioid receptor kappa 1 using [125I]-D-Pro10-dynorphin A[1-11] as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.48E+3nMAssay Description:Binding affinity against cloned human Opioid receptor mu 1 using [125I]FK33824 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligandMore data for this Ligand-Target Pair