BDBM50093227 CHEMBL3586608
SMILES Cl.CN(Cc1ccccc1)Cc1ccc(COc2ccc3c(CO)cc(=O)oc3c2)cc1
InChI Key InChIKey=USTALMYDYGSTPY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 12 hits for monomerid = 50093227
Affinity DataKi: 100nMAssay Description:Mixed type inhibition of electric eel AChE by Lineweaver-Burk plotMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Swedish Defence Research Agency
Curated by ChEMBL
Swedish Defence Research Agency
Curated by ChEMBL
Affinity DataKi: 4.50E+3nMAssay Description:Tight binding inhibition of recombinant human MAO-B expressed in Pichia pastoris assessed as inhibition constant using benzylamine as substrate at 10...More data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of rat brain MAO-B using kynuramine substrate in rat mitochondrial substrate by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of electric eel AChE by spectrophotometric Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of recombinant mouse AChE expressed in human HEK293F cells using acetylthiocholine iodide as substrate by spectrophotometric Ellman's meth...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Swedish Defence Research Agency
Curated by ChEMBL
Swedish Defence Research Agency
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine substrate by spectrophotometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant AChE by spectrophotometric Ellman's methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Swedish Defence Research Agency
Curated by ChEMBL
Swedish Defence Research Agency
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human MAO-B expressed in Pichia pastoris using kynuramine as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human AChE by spectrophotometric Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of equine serum BuChE by spectrophotometric Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of human serum BuChE by spectrophotometric Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine substrate by spectrophotometric assayMore data for this Ligand-Target Pair