BDBM50094688 2-(furan-2-yl)-8-isopentyl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine::2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-ylamine::CHEMBL315150
SMILES CC(C)CCn1cc2c(n1)nc(N)n1nc(nc21)-c1ccco1
InChI Key InChIKey=NXSARBYAOXIQJA-UHFFFAOYSA-N
Data 14 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 14 hits for monomerid = 50094688
Affinity DataKi: 0.780nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Displacement of [3H]-SCH- 58261 from human adenosine A2A receptor expressed in CHO cells; range 0.60-1.00More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of [3H]-CGS- 21680 binding to Adenosine A2A receptor in rat striatal homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-DPCPX from human adenosine A1 receptor expressed in CHO cells; range 1.72-2.36More data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Inhibition of [3H]-CHA binding to Adenosine A1 receptor in rat whole brain homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]-CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A2b receptor expressed in CHO cells; range 7.4-11.3More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Displacement of [3H]-MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells; range 664-738More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.08E+5nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair