BDBM50098694 3-[(Benzyl-ethyl-amino)-methyl]-4-phenyl-quinoline-2-carboxylic acid diethylamide::CHEMBL6645

SMILES CCN(Cc1ccccc1)Cc1c(nc2ccccc2c1-c1ccccc1)C(=O)N(CC)CC

InChI Key InChIKey=GXAQSWNUEMPKQP-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50098694   

TargetTranslocator protein(Rat)
Rottapharm Biotech

Curated by ChEMBL
LigandPNGBDBM50098694(3-[(Benzyl-ethyl-amino)-methyl]-4-phenyl-quinoline...)
Affinity DataIC50: 4.10nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat brain cortex membrane incubated for 120 mins by liquid scintillation spectrometer methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTranslocator protein(Rat)
Rottapharm Biotech

Curated by ChEMBL
LigandPNGBDBM50098694(3-[(Benzyl-ethyl-amino)-methyl]-4-phenyl-quinoline...)
Affinity DataIC50: 4.10nMAssay Description:Test in vitro, for potential ability to displace [3H]1 from PBR in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed