BDBM50101665 5-Acetyl-4-{4-[4-(5-chloro-2-methoxy-phenyl)-piperazin-1-yl]-butylamino}-2,6-dimethyl-2H-pyridazin-3-one::CHEMBL420959
SMILES COc1ccc(Cl)cc1N1CCN(CCCCNc2c(C(C)=O)c(C)nn(C)c2=O)CC1
InChI Key InChIKey=LQABNCQTZIOQJK-UHFFFAOYSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50101665
Target5-hydroxytryptamine receptor 1A(Human)
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 1.39nMAssay Description:Binding affinity towards human cloned 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Human)
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 2.99nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Human)
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 5.96nMAssay Description:Binding affinity towards human cloned alpha1d-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Human)
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Istituto Chimico Farmaceutico E Tossicologico
Curated by ChEMBL
Affinity DataKi: 49.1nMAssay Description:Binding affinity towards human cloned alpha1B-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair