BDBM50117183 2,3,7,11b-Tetrahydro-1H-dibenzo[de,h]isoquinoline-8,9-diol::CHEMBL123642::Dinapsoline, (S)(-)

SMILES Oc1ccc2[C@H]3CNCc4cccc(Cc2c1O)c34

InChI Key InChIKey=ZQTSNGJHMUKLOM-UHFFFAOYSA-N

Data  2 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50117183   

TargetD(2) dopamine receptor(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50117183(CHEMBL123642 | Dinapsoline, (S)(-) | 2,3,7,11b-Tet...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibition of [125I]7-OH-PIPAT binding to Dopamine receptor D2 of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50117183(CHEMBL123642 | Dinapsoline, (S)(-) | 2,3,7,11b-Tet...)
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50117183(CHEMBL123642 | Dinapsoline, (S)(-) | 2,3,7,11b-Tet...)
Affinity DataIC50: 5.30E+3nMAssay Description:In vitro inhibition of [125I]SCH-23982 binding to Dopamine receptor D1 of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50117183(CHEMBL123642 | Dinapsoline, (S)(-) | 2,3,7,11b-Tet...)
Affinity DataKi:  5.30E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed