BDBM50122343 (S)-3-[4-(2-Diphenylamino-ethoxy)-phenyl]-2-ethoxy-propionic acid::CHEMBL86657

SMILES CCO[C@@H](Cc1ccc(OCCN(c2ccccc2)c2ccccc2)cc1)C(O)=O

InChI Key InChIKey=KASBLUIPHVTDNF-UHFFFAOYSA-N

Data  8 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50122343   

LigandPNGBDBM50122343((S)-3-[4-(2-Diphenylamino-ethoxy)-phenyl]-2-ethoxy...)
Affinity DataEC50:  3.30E+3nMAssay Description:Transactivation of GAL4-fused Homo sapiens (human) PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2014
Entry Details Article

LigandPNGBDBM50122343((S)-3-[4-(2-Diphenylamino-ethoxy)-phenyl]-2-ethoxy...)
Affinity DataEC50:  3.30E+3nMAssay Description:In vitro activation of human peroxisome proliferator activated receptor gamma (PPAR gamma)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50122343((S)-3-[4-(2-Diphenylamino-ethoxy)-phenyl]-2-ethoxy...)
Affinity DataEC50:  3.30E+3nMAssay Description:Transactivation of GAL4-fused Homo sapiens (human) PPARgamma DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2014
Entry Details Article

LigandPNGBDBM50122343((S)-3-[4-(2-Diphenylamino-ethoxy)-phenyl]-2-ethoxy...)
Affinity DataEC50:  3.31E+3nMAssay Description:Transactivation of Homo sapiens (human) PPARgamma assessed as luciferase activity by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

LigandPNGBDBM50122343((S)-3-[4-(2-Diphenylamino-ethoxy)-phenyl]-2-ethoxy...)
Affinity DataEC50:  4.47E+3nMAssay Description:Transactivation of Homo sapiens (human) PPARalpha assessed as luciferase activity by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

LigandPNGBDBM50122343((S)-3-[4-(2-Diphenylamino-ethoxy)-phenyl]-2-ethoxy...)
Affinity DataEC50:  4.50E+3nMAssay Description:Transactivation of GAL4-fused Homo sapiens (human) PPARalpha DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2014
Entry Details Article

LigandPNGBDBM50122343((S)-3-[4-(2-Diphenylamino-ethoxy)-phenyl]-2-ethoxy...)
Affinity DataEC50:  4.50E+3nMAssay Description:In vitro activation of human peroxisome proliferator activated receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50122343((S)-3-[4-(2-Diphenylamino-ethoxy)-phenyl]-2-ethoxy...)
Affinity DataEC50:  4.50E+3nMAssay Description:Transactivation of GAL4-fused Homo sapiens (human) PPARalpha DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2014
Entry Details Article