BDBM50129149 5-[1,3]Dithian-2-ylidene-9-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene::CHEMBL65929
SMILES [#6]-[#6]-1=[#6]C([#6])([#6])[#7]-c2ccc3-c4cc(F)ccc4-[#8]\[#6](=[#6]-4/[#16]-[#6]-[#6]-[#6]-[#16]-4)-c3c-12
InChI Key InChIKey=NTCBYBDADUSXSB-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50129149
Affinity DataKi: 6.30nMAssay Description:Binding affinity to human progesterone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 146nMAssay Description:Antagonist activity at glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10nMAssay Description:Effective concentration for agonist activity towards human progesterone receptor (hPR) using the cotransfection assay in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:Inhibitory concentration for antagonistic activity towards human progesterone receptor (hPR) using the cotransfection assay in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 681nMAssay Description:Antagonist activity at mineralocorticoid receptor (hMR)More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Antagonist activity against human Androgen receptorMore data for this Ligand-Target Pair