BDBM50130336 CHEMBL3633296

SMILES CC(C)c1cccc(NC(=O)Nc2cccc(c2)-c2cccc3[nH]nc(N)c23)c1

InChI Key InChIKey=PNJKZZZAABVQNH-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50130336   

TargetVascular endothelial growth factor receptor 2(Human)
The First Affiliated Hospital of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50130336(CHEMBL3633296)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of VEGFR-2 (unknown origin) after 1 hr by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
The First Affiliated Hospital of Xi'An Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50130336(CHEMBL3633296)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged VEGFR2 (789 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly (4:1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed