BDBM50134847 4-(3-Ethyl-1-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-g]quinazolin-8-yl)-piperazine-1-carbothioic acid benzylamide::CHEMBL434262

SMILES CCn1c2cc3ncnc(N4CCN(CC4)C(=S)NCc4ccccc4)c3cc2n(C)c1=O

InChI Key InChIKey=HFCYEHKOQAJLRK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50134847   

TargetPlatelet-derived growth factor receptor beta(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50134847(4-(3-Ethyl-1-methyl-2-oxo-2,3-dihydro-1H-imidazo[4...)
Affinity DataIC50: 140nMAssay Description:Inhibition of platelet-derived growth factor receptor beta phosphorylation was measured in intact cells using a two-site enzyme linked immunosorbent ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed