BDBM50138763 (S)-2-({2'-Methyl-5-[2-(3-methyl-3H-imidazol-4-yl)-acetylamino]-biphenyl-2-carbonyl}-amino)-4-methylsulfanyl-butyric acid::CHEMBL138192

SMILES CSCC[C@H](NC(=O)c1ccc(NC(=O)Cc2cncn2C)cc1-c1ccccc1C)C(O)=O

InChI Key InChIKey=DDTGELIOCFLYLI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50138763   

TargetDimer of Protein farnesyltransferase subunit beta(Human)
Yale University

Curated by ChEMBL
LigandPNGBDBM50138763((S)-2-({2'-Methyl-5-[2-(3-methyl-3H-imidazol-4-yl)...)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of Trypanosoma brucei protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed