BDBM50155966 4-(2-Bromo-4-isopropyl-phenyl)-8-(ethyl-furan-2-ylmethyl-amino)-6-methyl-3,4-dihydro-1H-pyrido[2,3-b]pyrazin-2-one::CHEMBL188858

SMILES CCN(Cc1ccco1)c1cc(C)nc2N(CC(=O)Nc12)c1ccc(cc1Br)C(C)C

InChI Key InChIKey=NYZRYJPGNDZZEO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50155966   

TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50155966(4-(2-Bromo-4-isopropyl-phenyl)-8-(ethyl-furan-2-yl...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [125I]ovine-CRF binding to corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed