BDBM50158564 1-(5-Chloro-2-hydroxy-phenyl)-3-(3-trifluoromethyl-phenyl)-urea::1-(5-chloro-2-hydroxyphenyl)-3-(3-trifluoromethylphenyl)urea::CHEMBL33891

SMILES Oc1ccc(Cl)cc1NC(=O)Nc1cccc(c1)C(F)(F)F

InChI Key InChIKey=KRHJDJMOIKRPNN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50158564   

TargetGlutamate receptor ionotropic, kainate 1(Human)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50158564(1-(5-chloro-2-hydroxyphenyl)-3-(3-trifluoromethylp...)
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at human homomeric GluR5 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed