BDBM50158567 2-[2-(3-bromophenylamino)-3,4-dioxocyclobut-1-enylamino]-4-chlorobenzoic acid::CHEMBL224785

SMILES OC(=O)c1ccc(Cl)cc1Nc1c(Nc2cccc(Br)c2)c(=O)c1=O

InChI Key InChIKey=QYFRNJPTCNVDDB-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50158567   

TargetGlutamate receptor ionotropic, kainate 1(Human)
The Danish University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50158567(2-[2-(3-bromophenylamino)-3,4-dioxocyclobut-1-enyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at human homomeric GluR5 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed