BDBM50163218 4-(3-Methyl-pyridin-2-yl)-piperazine-1-carboxylic acid (4-chloro-phenyl)-amide::CHEMBL369647

SMILES Cc1cccnc1N1CCN(CC1)C(=O)Nc1ccc(Cl)cc1

InChI Key InChIKey=IMQPEOBFOGPGNI-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50163218   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50163218(4-(3-Methyl-pyridin-2-yl)-piperazine-1-carboxylic ...)
Affinity DataIC50: 113nMAssay Description:Inhibition of human transient receptor potential vanilloid 1 receptor (n=4)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50163218(4-(3-Methyl-pyridin-2-yl)-piperazine-1-carboxylic ...)
Affinity DataIC50: 409nMAssay Description:Inhibition of rat transient receptor potential vanilloid 1 receptor (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed