BDBM50168703 1-((R)-2-Amino-2-phenyl-ethyl)-3-(2-fluoro-3-methoxy-phenyl)-5-(2-trifluoromethoxy-benzyl)-[1,3,5]triazinane-2,4,6-trione::CHEMBL425523
SMILES COc1cccc(c1F)-n1c(=O)n(C[C@H](N)c2ccccc2)c(=O)n(Cc2ccccc2OC(F)(F)F)c1=O
InChI Key InChIKey=LJJACIKIUOHOLD-SFHVURJKSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50168703
Affinity DataKi: 18nMAssay Description:In vitro ability to inhibit des-Gly[125I-Tyr, DLeu, NMeLeu,Pro-NEt]-GnRH radioligand binding to the cloned human GnRH receptor stably expressed in HE...More data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Inhibition constant against monkey GnRH receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.40E+3nMAssay Description:Inhibition constant against rat GnRH receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of human GnRH receptor stimulated inositol phosphate accumulation in RBL cellsMore data for this Ligand-Target Pair