BDBM50172920 3-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(piperidin-4-yl)benzamide::3-[6-(2-Chloro-phenylamino)-1H-indazol-3-yl]-N-piperidin-4-yl-benzamide::CHEMBL194806

SMILES Clc1ccccc1Nc1ccc2c(n[nH]c2c1)-c1cccc(c1)C(=O)NC1CCNCC1

InChI Key InChIKey=VKTAENBLRPMXKK-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50172920   

TargetMitogen-activated protein kinase 10(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50172920(3-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(pip...)
Affinity DataIC50: 1.26nMAssay Description:Inhibition of JNK3 by high throughput screeningMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50172920(3-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(pip...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against c-Jun N-terminal kinase 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50172920(3-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(pip...)
Affinity DataIC50: 3.98nMAssay Description:Inhibition of p38alpha by high throughput screeningMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50172920(3-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(pip...)
Affinity DataIC50: 4.40nMAssay Description:Inhibitory concentration against Mitogen-activated protein kinase p38 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50172920(3-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(pip...)
Affinity DataIC50: 71nMAssay Description:Inhibitory concentration against c-Jun N-terminal kinase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Astrazeneca R&D SöDertäLje

Curated by ChEMBL
LigandPNGBDBM50172920(3-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(pip...)
Affinity DataIC50: 79.4nMAssay Description:Inhibition of JNK1 by high throughput screeningMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed