BDBM50174879 CHEMBL370665::X2-Apc-DPhe-Arg-Trp-Z4-NH2

SMILES CCCCNC(=O)N[C@@]1(CC[C@@H](CC1)c1ccccc1)C(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCCC(N)=O

InChI Key InChIKey=FWAGLFKWEVDSRV-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50174879   

TargetMelanocortin receptor 4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50174879(X2-Apc-DPhe-Arg-Trp-Z4-NH2 | CHEMBL370665)
Affinity DataEC50:  2nMAssay Description:Agonist activity in HEK293 cells transfected with human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed