BDBM50177564 CHEMBL380540::N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1-(2-fluorophenyl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-1,1-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
SMILES CCN(CC)CC(N1CCN(CC1)C(=O)[C@@H](Cc1ccc(Cl)cc1)NC(=O)C1Cc2ccccc2C(C)(C)N1)c1ccccc1F
InChI Key InChIKey=HEILVIDOVAHKRM-QVGGVDQBSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50177564
Affinity DataKi: 5.80nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cellMore data for this Ligand-Target Pair