BDBM50185544 2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(1-methylpiperidin-4-yl)-1H-indole::CHEMBL379284

SMILES CN1CCC(CC1)c1cccc2[nH]c(cc12)-c1nc(CCc2ccc(Cl)cc2)no1

InChI Key InChIKey=XRRSGVAKNLABMJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50185544   

TargetNociceptin receptor(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185544(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(...)
Affinity DataIC50: 62nMAssay Description:Displacement of [125I][Tyr14]N/OFQ from ORL1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50185544(2-(3-(4-chlorophenethyl)-1,2,4-oxadiazol-5-yl)-4-(...)
Affinity DataIC50: 899nMAssay Description:Antagonist activity against ORL1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed