BDBM50186343 CHEMBL3824187

SMILES CCc1cnc(nc1)N1CCC(CC1)n1ncc2cc(ncc12)-c1ccc(cc1)S(C)(=O)=O

InChI Key InChIKey=UGNWKIREOVBGOL-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50186343   

TargetGlucose-dependent insulinotropic receptor(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50186343(CHEMBL3824187)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR119 expressed in Flp-In-T-Rex-HEK293 cells assessed as stimulation of cAMP level measured after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50186343(CHEMBL3824187)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR119 expressed in Flp-In-T-Rex-HEK293 cells after 30 mins by cAMP accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2017
Entry Details Article
PubMed