BDBM50191267 CHEMBL376703::H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys]-Thr-NH2

SMILES C[C@@H](O)[C@H](NC(=O)[C@@H]1CSSC[C@H](NC(=O)[C@H](N)Cc2ccccc2)C(=O)N[C@@H](C)C(=O)N[C@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]([C@@H](C)O)C(=O)N1)C(N)=O

InChI Key InChIKey=DNIBTKHTGSPUNA-RHSAGAAYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50191267   

TargetSomatostatin receptor type 3(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50:  543nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50191267(CHEMBL376703 | H-D-Phe-c[Cys-Ala-D-Trp-Lys-Thr-Cys...)
Affinity DataIC50:  158nMAssay Description:Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed